A facile aminocyclization for the synthesis of pyrrolidine and piperidine derivatives.
نویسندگان
چکیده
Bromination of an isolated double bond followed by aminocyclization furnishes a highly stereoselective protocol for the intramolecular formation of pyrrolidine and piperidine ring containing subunits that are presented in numerous biologically active natural products.
منابع مشابه
SYNTHESIS AND CHARACTERIZATION OF AMINE(CHLOR0)COBALOXIME DERIVATIVES. APPROXIMATE VALUES OF THE ANGULAROVERLAP PARAMETER, ?, FOR THE COORDINATED AMINES
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ورودعنوان ژورنال:
- Chemical communications
دوره 15 شماره
صفحات -
تاریخ انتشار 2003